Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 5951
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102430(US8536173, 5)
Affinity DataIC50:  11nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102428(US8536173, 3)
Affinity DataIC50:  21nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102429(US8536173, 4)
Affinity DataIC50:  23nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102434(US8536173, 9)
Affinity DataIC50:  31nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102427(US8536173, 2)
Affinity DataIC50:  32nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102432(US8536173, 7)
Affinity DataIC50:  45nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102431(US8536173, 6)
Affinity DataIC50:  57nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102426(US8536173, 1)
Affinity DataIC50:  68nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM102433(US8536173, 8)
Affinity DataIC50:  204nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM8528(US8536173, 10)
Affinity DataIC50:  720nMAssay Description:The measuring of the inhibitory activity in vitro of compounds in this invention on the enzyme 11bHSD1 using a Scintillation Proximity Assay (SPA) in...More data for this Ligand-Target Pair
In DepthDetails US Patent