Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 6487
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131882(US8835444, 5.27)
Affinity DataIC50:  13nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131876(US8835444, 5.1)
Affinity DataIC50:  21nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131881(US8835444, 5.26)
Affinity DataIC50:  22nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131860(US8835444, 1.8)
Affinity DataIC50:  35nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131875(US8835444, 4.6)
Affinity DataIC50:  40nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131883(US8835444, 5.29)
Affinity DataIC50:  49nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131872(US8835444, 4.2)
Affinity DataIC50:  59nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131878(US8835444, 5.11)
Affinity DataIC50:  67nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131871(US8835444, 4.1)
Affinity DataIC50:  82nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM9237(US8835444, 4.3 | US8835444, 4.8)
Affinity DataIC50:  88nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131880(US8835444, 5.21)
Affinity DataIC50:  95nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131877(US8835444, 5.8)
Affinity DataIC50:  126nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131863(US8835444, 2.4)
Affinity DataIC50:  131nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131879(US8835444, 5.17)
Affinity DataIC50:  132nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131858(US8835444, 1.1)
Affinity DataIC50:  134nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131869(US8835444, 3.6)
Affinity DataIC50:  142nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131867(US8835444, 2.16)
Affinity DataIC50:  147nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131861(US8835444, 2.0)
Affinity DataIC50:  160nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131864(US8835444, 2.13)
Affinity DataIC50:  167nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131866(US8835444, 2.15)
Affinity DataIC50:  170nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131868(US8835444, 3.3)
Affinity DataIC50:  180nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131865(US8835444, 2.14)
Affinity DataIC50:  214nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM9227(US8835444, 2.1)
Affinity DataIC50:  256nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM9237(US8835444, 4.3 | US8835444, 4.8)
Affinity DataIC50:  262nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131862(US8835444, 2.3)
Affinity DataIC50:  318nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131870(US8835444, 3.17)
Affinity DataIC50:  634nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131874(US8835444, 4.5)
Affinity DataIC50:  665nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131860(US8835444, 1.8)
Affinity DataIC50:  727nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131859(US8835444, 1.4)
Affinity DataIC50:  948nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131882(US8835444, 5.27)
Affinity DataIC50:  2.03E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131869(US8835444, 3.6)
Affinity DataIC50:  3.74E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131868(US8835444, 3.3)
Affinity DataIC50:  4.63E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131880(US8835444, 5.21)
Affinity DataIC50:  4.85E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131858(US8835444, 1.1)
Affinity DataIC50:  4.88E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131863(US8835444, 2.4)
Affinity DataIC50:  4.94E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM131873(US8835444, 4.4)
Affinity DataIC50:  6.96E+3nMAssay Description:Chinese hamster ovary (CHO) cells expressing either the human or rat recombinant CRF-1 or human CRF-2alpha (Chen et al, Proc Natl Acad Sci USA 90, 89...More data for this Ligand-Target Pair
In DepthDetails US Patent