Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 6505
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358213(CHEMBL1922219 | US8846696, (2R3S)-3-{9-Isopropyl-6...)
Affinity DataIC50:  30nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358211(CHEMBL1922212 | US8846696, (3S)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  70nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358212(CHEMBL1922218 | US8846696, (2S3R)-3-{9-Isopropyl-6...)
Affinity DataIC50:  90nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358235(CHEMBL1922209 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  110nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358210(CHEMBL1922123 | US8846696, (3R)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  200nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358221(CHEMBL1922120 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  220nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358237(CHEMBL1922211 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  390nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358212(CHEMBL1922218 | US8846696, (2S3R)-3-{9-Isopropyl-6...)
Affinity DataIC50:  500nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358222(CHEMBL1922121 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  690nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358223(CHEMBL1922122 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  1.00E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358221(CHEMBL1922120 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  1.10E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358236(CHEMBL1922210 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.10E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358213(CHEMBL1922219 | US8846696, (2R3S)-3-{9-Isopropyl-6...)
Affinity DataIC50:  1.30E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358235(CHEMBL1922209 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.50E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358223(CHEMBL1922122 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  1.60E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358213(CHEMBL1922219 | US8846696, (2R3S)-3-{9-Isopropyl-6...)
Affinity DataIC50:  2.20E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358222(CHEMBL1922121 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.20E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358211(CHEMBL1922212 | US8846696, (3S)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  2.50E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358210(CHEMBL1922123 | US8846696, (3R)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  3.10E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358237(CHEMBL1922211 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  3.50E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358236(CHEMBL1922210 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  3.50E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358211(CHEMBL1922212 | US8846696, (3S)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  4.40E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358212(CHEMBL1922218 | US8846696, (2S3R)-3-{9-Isopropyl-6...)
Affinity DataIC50:  4.90E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358210(CHEMBL1922123 | US8846696, (3R)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  6.20E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358213(CHEMBL1922219 | US8846696, (2R3S)-3-{9-Isopropyl-6...)
Affinity DataIC50:  6.80E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358210(CHEMBL1922123 | US8846696, (3R)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  7.50E+3nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358235(CHEMBL1922209 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358221(CHEMBL1922120 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  1.20E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358211(CHEMBL1922212 | US8846696, (3S)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  1.20E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358237(CHEMBL1922211 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.30E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358235(CHEMBL1922209 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.30E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358212(CHEMBL1922218 | US8846696, (2S3R)-3-{9-Isopropyl-6...)
Affinity DataIC50:  1.40E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358235(CHEMBL1922209 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  1.70E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358222(CHEMBL1922121 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.00E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358213(CHEMBL1922219 | US8846696, (2R3S)-3-{9-Isopropyl-6...)
Affinity DataIC50:  2.00E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358222(CHEMBL1922121 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358237(CHEMBL1922211 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  2.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358236(CHEMBL1922210 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  2.20E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358212(CHEMBL1922218 | US8846696, (2S3R)-3-{9-Isopropyl-6...)
Affinity DataIC50:  2.30E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358223(CHEMBL1922122 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.30E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358237(CHEMBL1922211 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  2.30E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358223(CHEMBL1922122 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.40E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358221(CHEMBL1922120 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  2.50E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358236(CHEMBL1922210 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  3.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358211(CHEMBL1922212 | US8846696, (3S)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  3.50E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358221(CHEMBL1922120 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  3.70E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358223(CHEMBL1922122 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  5.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358236(CHEMBL1922210 | US8846696, (3RS,4S)-4-{9-Isopropyl...)
Affinity DataIC50:  6.70E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358210(CHEMBL1922123 | US8846696, (3R)-3-{9-Isopropyl-6-[...)
Affinity DataIC50:  9.10E+4nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cyclacel

US Patent
LigandPNGBDBM50358222(CHEMBL1922121 | US8846696, (3RS,4R)-4-{9-Isopropyl...)
Affinity DataIC50:  1.11E+5nMpH: 7.4Assay Description:The compounds from the examples below were investigated for their CDK2/cyclin E, CDK1/cyclin B, CDK4/cyclin D1 and CDK7/cyclin H, ERK-2, and PKA inhi...More data for this Ligand-Target Pair
In DepthDetails US Patent
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