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Found 71 Enz. Inhib. hit(s) with all data for entry = 6543
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138193(US8877798, Table 3, Structure 39)
Affinity DataKi:  6nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138157(US8877798, Table 3, Structure 3)
Affinity DataKi:  13nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138155(US8877798, Table 3, Structure 1)
Affinity DataKi:  16nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138167(US8877798, Table 3, Structure 13)
Affinity DataKi:  25nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138157(US8877798, Table 3, Structure 3)
Affinity DataKi:  32nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138166(US8877798, Table 3, Structure 12)
Affinity DataKi:  39nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138158(US8877798, Table 3, Structure 4)
Affinity DataKi:  46nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138156(US8877798, Table 3, Structure 2)
Affinity DataKi:  62nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138193(US8877798, Table 3, Structure 39)
Affinity DataKi:  68nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138168(US8877798, Table 3, Structure 14)
Affinity DataKi:  72nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138155(US8877798, Table 3, Structure 1)
Affinity DataKi:  81nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138157(US8877798, Table 3, Structure 3)
Affinity DataKi:  88nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138155(US8877798, Table 3, Structure 1)
Affinity DataKi:  105nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138158(US8877798, Table 3, Structure 4)
Affinity DataKi:  113nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138166(US8877798, Table 3, Structure 12)
Affinity DataKi:  124nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138156(US8877798, Table 3, Structure 2)
Affinity DataKi:  125nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138168(US8877798, Table 3, Structure 14)
Affinity DataKi:  132nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138161(US8877798, Table 3, Structure 7)
Affinity DataKi:  170nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138175(US8877798, Table 3, Structure 21)
Affinity DataKi:  190nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138164(US8877798, Table 3, Structure 10)
Affinity DataKi:  215nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138160(US8877798, Table 3, Structure 6)
Affinity DataKi:  220nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138173(US8877798, Table 3, Structure 19)
Affinity DataKi:  230nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138162(US8877798, Table 3, Structure 8)
Affinity DataKi:  240nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138159(US8877798, Table 3, Structure 5)
Affinity DataKi:  250nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138184(US8877798, Table 3, Structure 30)
Affinity DataKi:  260nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138184(US8877798, Table 3, Structure 30)
Affinity DataKi:  270nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138167(US8877798, Table 3, Structure 13)
Affinity DataKi:  330nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138175(US8877798, Table 3, Structure 21)
Affinity DataKi:  350nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138163(US8877798, Table 3, Structure 9)
Affinity DataKi:  395nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138170(US8877798, Table 3, Structure 16)
Affinity DataKi:  420nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138156(US8877798, Table 3, Structure 2)
Affinity DataKi:  490nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138180(US8877798, Table 3, Structure 26)
Affinity DataKi:  500nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138167(US8877798, Table 3, Structure 13)
Affinity DataKi:  510nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138193(US8877798, Table 3, Structure 39)
Affinity DataKi:  520nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138181(US8877798, Table 3, Structure 27)
Affinity DataKi:  540nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138158(US8877798, Table 3, Structure 4)
Affinity DataKi:  585nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138175(US8877798, Table 3, Structure 21)
Affinity DataKi:  640nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138173(US8877798, Table 3, Structure 19)
Affinity DataKi:  680nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138187(US8877798, Table 3, Structure 33)
Affinity DataKi:  710nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138170(US8877798, Table 3, Structure 16)
Affinity DataKi:  800nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138166(US8877798, Table 3, Structure 12)
Affinity DataKi:  827nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138184(US8877798, Table 3, Structure 30)
Affinity DataKi:  830nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138181(US8877798, Table 3, Structure 27)
Affinity DataKi:  920nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138172(US8877798, Table 3, Structure 18)
Affinity DataKi:  990nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138161(US8877798, Table 3, Structure 7)
Affinity DataKi:  1.07E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138165(US8877798, Table 3, Structure 11)
Affinity DataKi:  1.10E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138164(US8877798, Table 3, Structure 10)
Affinity DataKi:  1.10E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138172(US8877798, Table 3, Structure 18)
Affinity DataKi:  1.60E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138159(US8877798, Table 3, Structure 5)
Affinity DataKi:  1.67E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransporter(Rattus norvegicus (rat))
Neurovance

US Patent
LigandPNGBDBM138173(US8877798, Table 3, Structure 19)
Affinity DataKi:  1.70E+3nMAssay Description:Binding assay using NET, DAT and SERT enzyme.More data for this Ligand-Target Pair
In DepthDetails US Patent
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