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Found 7 Enz. Inhib. hit(s) with all data for entry = 6726
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150169(US8980887, Compound 13)
Affinity DataKi:  2.97nM ΔG°:  -49.5kJ/mole IC50:  6.99nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150168(US8980887, Compound 11)
Affinity DataKi:  6.66nM ΔG°:  -47.5kJ/mole IC50:  15.6nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150164(US8980887, Compound 1)
Affinity DataKi:  7.17nM ΔG°:  -47.3kJ/mole IC50:  16.9nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150166(US8980887, Compound 8)
Affinity DataKi:  9.34nM ΔG°:  -46.6kJ/mole IC50:  21.9nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150167(US8980887, Compound 10)
Affinity DataKi:  11.1nM ΔG°:  -46.2kJ/mole IC50:  26.1nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150170(US8980887, Compound 14)
Affinity DataKi:  38.7nM ΔG°:  -43.0kJ/mole IC50:  91.0nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranslocator protein(Rattus norvegicus (rat))
Toxicology Academy Of Military Medical Sciences P.L.A.

US Patent
LigandPNGBDBM150165(US8980887, Compound 7)
Affinity DataKi:  49.2nM ΔG°:  -42.4kJ/mole IC50:  116nMT: 2°CAssay Description:Competitive Binding Test of Drug to the Receptor (Rat Heart TSPO) and Radioligand (3H-PK11195): (1) tubes were placed in reaction condition of 30 C.(...More data for this Ligand-Target Pair
In DepthDetails US Patent