Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 6841
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153641(US8999982, Ref4)
Affinity DataIC50:  7.04E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153643(US8999982, Ref6)
Affinity DataIC50:  8.29E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153652(US8999982, 3-fluoro-4-((6-methoxy-7-(3- morpholino...)
Affinity DataIC50:  8.50E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153644(US8999982, Ref7)
Affinity DataIC50:  9.30E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153645(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153646(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)ani...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153647(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153648(US8999982, 3-chloro-4-((6,7- dimethoxyquinolin-4- ...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153649(US8999982, 5-((6,7-dimethoxyquinolin-4- yl)oxy)pyr...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153650(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153651(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153642(US8999982, Ref5)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153640(US8999982, Ref3)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153653(US8999982, tert-butyl 4-(((4-(4-amino-2- fluorophe...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM50317324(CHEMBL1087984 | N-(4-(6,7-dimethoxyquinolin-4-ylox...)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center

US Patent
LigandPNGBDBM153639(US8999982, Ref2)
Affinity DataIC50: >1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent