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Found 16 Enz. Inhib. hit(s) with all data for entry = 4085
TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM10515(5-(1,2-dithiolan-3-yl)pentanoic acid | CHEMBL33864...)
Affinity DataIC50:  201nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataIC50:  901nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM40324((4Z)-2-nitro-4-[(2-thiazolylhydrazo)methylidene]-1...)
Affinity DataIC50:  2.69E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM34334(MLS000055225 | N-[1,3-benzothiazol-2-yl(phenyl)pho...)
Affinity DataIC50:  3.10E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47028(3-(4-bromophenyl)sulfonyl-N-[(4-methylphenyl)methy...)
Affinity DataIC50:  3.27E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47027(2-(3-brosylpropanoylamino)benzoic acid methyl este...)
Affinity DataIC50:  3.33E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47024((2E,3E)-3-(3-methoxy-4-oxidanylidene-cyclohexa-2,5...)
Affinity DataIC50:  4.53E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM34849(6-fluoranyl-2-(2-methylphenyl)-1,2-benzothiazol-3-...)
Affinity DataIC50:  4.57E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47026((Z)-2-methyl-6-[(5R,10S,13R,14R,17R)-4,4,10,13,14-...)
Affinity DataIC50:  5.81E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47023(2-methyl-N-undecyl-3-furamide | 2-methyl-N-undecyl...)
Affinity DataIC50:  6.41E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM46667(2-phenyl-1,2-benzothiazol-3-one | 2-phenyl-1,2-ben...)
Affinity DataIC50:  6.80E+3nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM34709(MLS000567780 | N-(1-adamantyl)-2-(3-keto-1,2-benzo...)
Affinity DataIC50:  1.07E+4nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM43272(4-chloranyl-2-[(4-methoxyphenyl)carbonylamino]benz...)
Affinity DataIC50:  1.58E+4nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM29632(2-[2-(3-keto-1,2-benzothiazol-2-yl)thiazol-4-yl]ac...)
Affinity DataIC50:  3.66E+4nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM47025((4E)-4-[(5-butyl-2-thienyl)methylene]-3-phenyl-2-i...)
Affinity DataIC50: >1.00E+5nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
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TargetPhosphotransferase(Trypanosoma brucei)
University Of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM34960(2-(1,3-thiazol-2-yl)-1,2-benzothiazol-3-one | 2-(2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Excerpt from MH082340 application (Dr. James Morris, Clemson University) Trypanosoma brucei, the digenic protozoan parasite that causes African sleep...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay