Reaction Details Report a problem with these data
Target
Aurora kinase B [1-341]
Ligand
BDBM311130
Substrate
n/a
Meas. Tech.
Aurora B Kinase Test
IC50
50000±n/a nM
Citation
Hoffmann, M; Dahmann, G; Gnamm, C; Fandrick, DR; Scott, J; McCarthy, C Pyrazolyl-substituted heteroaryls and their use as medicaments US Patent US10155751 Publication Date 12/18/2018
More Info.:
Target
Name:
Aurora kinase B [1-341]
Synonyms:
AIK2 | AIM1 | AIRK2 | ARK2 | AURB (aa 1-341) | AURKB | AURKB_HUMAN | STK1 | STK12 | STK5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39070.43
Organism:
Homo sapiens (Human)
Description:
Q96GD4[1-341]
Residue:
341
Sequence:
MAQKENSYPWPYGRQTAPSGLSTLPQRVLRKEPVTPSALVLMSRSNVQPTAAPGQKVMENSSGTPDILTRHFTIDDFEIGRPLGKGKFGNVYLAREKKSHFIVALKVLFKSQIEKEGVEHQLRREIEIQAHLHHPNILRLYNYFYDRRRIYLILEYAPRGELYKELQKSCTFDEQRTATIMEELADALMYCHGKKVIHRDIKPENLLLGLKGELKIADFGWSVHAPSLRRKTMCGTLDYLPPEMIEGRMHNEKVDLWCIGVLCYELLVGNPPFESASHNETYRRIVKVDLKFPASVPMGAQDLISKLLRHNPSERLPLAQVSAHPWVRANSRRVLPPSALQ