Reaction Details Report a problem with these data
Target
Somatostatin receptor type 5
Ligand
BDBM311927
Substrate
n/a
Meas. Tech.
Radiogland Binding Assays
Ki
>8079±n/a nM
Citation
 Giovannini, R; Cui, Y; Doods, H; Ferrara, M; Just, S; Kuelzer, R; Lingard, I; Mazzaferro, R; Rudolf, K Somatostatin receptor subtype 4 (SSTR4) agonists US Patent  US10166214 Publication Date 1/1/2019 
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL
  
Inhibitor
Name:
BDBM311927
Synonyms:
US10166214, Example 63 | US10675268, Example 63 | US9789082, Example 63
Type:
Small organic molecule
Emp. Form.:
C16H20F3N3O2
Mol. Mass.:
343.3441
SMILES:
CC(C)(COc1cnccc1C(F)(F)F)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r|
Structure:
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