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TargetBromodomain-containing protein 2 Bromo 1 domain(BRD2 BD1)
LigandBDBM313795
Substrate/Competitorn/a
Meas. Tech.Binding Assay
IC50<100±n/a nM
Citation Burns, CGarnier, JSharp, PPFeutrill, JCuzzupe, A Benzodiazepines as bromodomain inhibitors US Patent US10167292 Publication Date 1/1/2019
More Info.:Get all data from this article,  Assay Method
 
Bromodomain-containing protein 2 Bromo 1 domain(BRD2 BD1)
Name:Bromodomain-containing protein 2 Bromo 1 domain(BRD2 BD1)
Synonyms:n/a
Type:n/a
Mol. Mass.:8836.08
Organism:Homo sapiens (Human)
Description:BD1 (91-163 aa) of P25440
Residue:73
Sequence:
WKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFT
NCYIYNKPTDDIV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM313795
NameBDBM313795
Synonyms:US10167292, Example 39
TypeSmall organic molecule
Emp. Form.C26H24ClN5O
Mol. Mass.457.955
SMILESC[C@@H](NC(=O)c1ccc2-c3c(C)nnn3CCN(c3ccc(Cl)cc3)c2c1)c1ccccc1 |r|
Structure
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n/a