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TargetPeroxisome proliferator-activated receptor delta
LigandBDBM323614
Substrate/Competitorn/a
Meas. Tech.Luciferase Assay
EC50 5544±n/a nM
Citation Downes, MEvans, RKluge, ALagu, BMiura, MPanigrahi, SKPatane, MSamajdar, SSenaiar, RTakahashi, T PPAR agonists, compounds, pharmaceutical compositions, and methods of use thereof US Patent US10188627 Publication Date 1/29/2019
More Info.:Get all data from this article,  Assay Method
 
Peroxisome proliferator-activated receptor delta
Name:Peroxisome proliferator-activated receptor
Synonyms:NR1C2 | NUC1 | NUCI | Nuclear hormone receptor 1 | Nuclear receptor subfamily 1 group C member 2 | PPAR delta | PPAR-beta | PPARB | PPARD | Peroxisome proliferator-activated receptor beta
Type:Enzyme
Mol. Mass.:49910.45
Organism:Homo sapiens (Human)
Description:Q03181
Residue:441
Sequence:
MEQPQEEAPEVREEEEKEEVAEAEGAPELNGGPQHALPSSSYTDLSRSSSPPSLLDQLQM
GCDGASCGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCERSCKIQKK
NRNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTANEGSQYNPQVADLKAFSK
HIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKE
ISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNK
DGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGD
RPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRI
KKTETETSLHPLLQEIYKDMY
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  Blast E-value cutoff:
BDBM323614
NameBDBM323614
Synonyms:Synthesis of 6-(2-((N,2-dimethylbenzofuran-5-carboxamido)methyl)phenoxy)-2,2-dimethylhexanoic acid | US10188627, Compound 8z
TypeSmall organic molecule
Emp. Form.C26H31NO5
Mol. Mass.437.528
SMILESCN(Cc1ccccc1OCCCCC(C)(C)C(O)=O)C(=O)c1ccc2oc(C)cc2c1
Structure
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n/a