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Targetb-raf
LigandBDBM205017
Substrate/Competitorn/a
Meas. Tech.Homogeneous Time-Resolved Fluorescence (HTRF) assay
IC50<500±0 nM
Citation Xiao, DLi, JZhu, YHu, YWang, HWang, ZWang, ZWei, YSun, YWu, QZhang, HPeng, YKong, FSun, YLuo, HHan, Y Kinase modulating compounds, compositions containing the same and use thereof US Patent US9550781 Publication Date 1/24/2017
More Info.:Get all data from this article,  Assay Method
 
b-raf
Name:SRC2-3 peptide
Synonyms:Human nuclear receptor coactivator 2 (residues 740-753)
Type:fluorescent labeled peptide
Mol. Mass.:1808.04
Organism:n/a
Description:n/a
Residue:15
Sequence:
CKENALLRYLLDKDD
 
BDBM205017
NameBDBM205017
Synonyms:US9550781, 14 | n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difluorophenyl)-3,4-difluorobenzenesulfonamide
TypeSmall organic molecule
Emp. Form.C22H13F4N7O2S
Mol. Mass.515.443
SMILESFc1ccc(cc1F)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Structure
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