Reaction Details Report a problem with these data
Target
Nuclear receptor coactivator 2 [740-753]
Ligand
BDBM228140
Substrate
n/a
Meas. Tech.
Competitive Binding Assay
IC50
7900±n/a nM
Citation
 Tanis, SP; Larsen, SD; Artman, III, GD; Parker, T PPAR-sparing compounds for the treatment of metabolic diseases US Patent  US9562012 Publication Date 2/7/2017 
Target
Name:
Nuclear receptor coactivator 2 [740-753]
Synonyms:
BHLHE75 | Human nuclear receptor coactivator 2 (aa 740-753) | NCOA2 | NCOA2_HUMAN | Nuclear receptor coactivator 2 (aa 740-753) | SRC2 | SRC2-3 peptide | TIF2
Type:
fluorescent labeled peptide
Mol. Mass.:
1704.90
Organism:
n/a
Description:
Q15596 aa 740-753
Residue:
14
Sequence:
KENALLRYLLDKDD
 
Inhibitor
Name:
BDBM228140
Synonyms:
(2s)-2-ethoxy-n-methoxy-3-{4-[(4-methoxypyridin-2-yl)methoxy]phenyl}propanamide hydrochloride (compound no. 5) | US9562012, 10
Type:
Small organic molecule
Emp. Form.:
C21H27NO7S
Mol. Mass.:
437.507
SMILES:
CCO[C@@H](Cc1ccc(OCCc2ccc(OS(C)(=O)=O)cc2)cc1)C(=O)NOC |r|
Structure:
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