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Target
AMSH-like protease
Ligand
BDBM401024
Substrate
n/a
Meas. Tech.
Biochemical Assay
IC50
25400±n/a nM
Citation
Deshaies, RJ; Li, J; Cohen, S; Perez, C; Ma, Y Inhibitors of RPN11 US Patent US10005735 Publication Date 6/26/2018
More Info.:
Target
Name:
AMSH-like protease
Synonyms:
AMSH-LP | AMSHLP | KIAA1373 | STALP_HUMAN | STAM-binding protein-like 1 (AMSH) | STAMBPL1
Type:
Protein
Mol. Mass.:
49789.14
Organism:
Homo sapiens (Human)
Description:
Q96FJ0
Residue:
436
Sequence:
MDQPFTVNSLKKLAAMPDHTDVSLSPEERVRALSKLGCNITISEDITPRRYFRSGVEMERMASVYLEEGNLENAFVLYNKFITLFVEKLPNHRDYQQCAVPEKQDIMKKLKEIAFPRTDELKNDLLKKYNVEYQEYLQSKNKYKAEILKKLEHQRLIEAERKRIAQMRQQQLESEQFLFFEDQLKKQELARGQMRSQQTSGLSEQIDGSALSCFSTHQNNSLLNVFADQPNKSDATNYASHSPPVNRALTPAATLSAVQNLVVEGLRCVVLPEDLCHKFLQLAESNTVRGIETCGILCGKLTHNEFTITHVIVPKQSAGPDYCDMENVEELFNVQDQHDLLTLGWIHTHPTQTAFLSSVDLHTHCSYQLMLPEAIAIVCSPKHKDTGIFRLTNAGMLEVSACKKKGFHPHTKEPRLFSICKHVLVKDIKIIVLDLR