Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37723
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
Ki
>40300±n/a nM
Comments
Extracted from aid = 520 and tid = 2
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37723
Synonyms:
2-cycloheptyl-3-keto-N-(3-pyridylmethyl)isoindoline-1-carboxamide | 2-cycloheptyl-3-oxidanylidene-N-(pyridin-3-ylmethyl)-1H-isoindole-1-carboxamide | 2-cycloheptyl-3-oxo-N-(3-pyridinylmethyl)-1H-isoindole-1-carboxamide | 2-cycloheptyl-3-oxo-N-(pyridin-3-ylmethyl)-1H-isoindole-1-carboxamide | 2-cycloheptyl-3-oxo-N-(pyridin-3-ylmethyl)isoindoline-1-carboxamide | MLS000087630 | SMR000023852 | cid_3241118
Type:
Small organic molecule
Emp. Form.:
C22H25N3O2
Mol. Mass.:
363.4528
SMILES:
O=C(NCc1cccnc1)C1N(C2CCCCCC2)C(=O)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: