Reaction Details Report a problem with these data
Target
Cathepsin G
Ligand
BDBM41380
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41380
Synonyms:
5-Methyl-pyrazine-2-carboxylic acid [2-(5-methyl-furan-2-yl)-phenyl]-amide | 5-methyl-N-[2-(5-methyl-2-furanyl)phenyl]-2-pyrazinecarboxamide | 5-methyl-N-[2-(5-methyl-2-furyl)phenyl]pyrazinamide | 5-methyl-N-[2-(5-methylfuran-2-yl)phenyl]pyrazine-2-carboxamide | MLS000076172 | SMR000000813 | cid_645091
Type:
Small organic molecule
Emp. Form.:
C17H15N3O2
Mol. Mass.:
293.3199
SMILES:
Cc1ccc(o1)-c1ccccc1NC(=O)c1cnc(C)cn1
Structure:
Search PDB for entries with ligand similarity: