Reaction Details Report a problem with these data
Target
Cathepsin G
Ligand
BDBM40847
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
2483.19±125.163 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM40847
Synonyms:
MLS000087424 | N-(2-phenylethyl)-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamide | N-(2-phenylethyl)-4,5-dihydronaphtho[2,1-d]isoxazole-3-carboxamide | N-phenethyl-4,5-dihydrobenz[g]indoxazene-3-carboxamide | SMR000023647 | cid_3240663
Type:
Small organic molecule
Emp. Form.:
C20H18N2O2
Mol. Mass.:
318.3691
SMILES:
O=C(NCCc1ccccc1)c1noc-2c1CCc1ccccc-21
Structure:
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