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Target
Cathepsin G
Ligand
BDBM38990
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM38990
Synonyms:
MLS000047015 | N-(3-fluoranyl-4-methyl-phenyl)-2-(3-methyl-4-oxidanylidene-phthalazin-1-yl)ethanamide | N-(3-fluoro-4-methyl-phenyl)-2-(4-keto-3-methyl-phthalazin-1-yl)acetamide | N-(3-fluoro-4-methylphenyl)-2-(3-methyl-4-oxo-1-phthalazinyl)acetamide | N-(3-fluoro-4-methylphenyl)-2-(3-methyl-4-oxo-3,4-dihydrophthalazin-1-yl)acetamide | N-(3-fluoro-4-methylphenyl)-2-(3-methyl-4-oxophthalazin-1-yl)acetamide | SMR000033026 | cid_2975205
Type:
Small organic molecule
Emp. Form.:
C18H16FN3O2
Mol. Mass.:
325.3369
SMILES:
Cc1ccc(NC(=O)Cc2nn(C)c(=O)c3ccccc23)cc1F
Structure:
Search PDB for entries with ligand similarity: