Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 1
Ligand
BDBM42495
Substrate
n/a
Meas. Tech.
Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism
IC50
5161±n/a nM
Citation
 PubChem, PC Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism PubChem Bioassay (2008)[AID] 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44399.07
Organism:
Homo sapiens (Human)
Description:
NPY-Y1 NPY1R HUMAN::P25929
Residue:
384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
  
Inhibitor
Name:
BDBM42495
Synonyms:
2-[2-[(benzylamino)methyl]phenoxy]-N-phenyl-acetamide;hydrochloride | 2-[2-[(benzylamino)methyl]phenoxy]-N-phenylacetamide;hydrochloride | 2-{2-[(benzylamino)methyl]phenoxy}-N-phenylacetamide hydrochloride | MLS000537927 | N-phenyl-2-[2-[[(phenylmethyl)amino]methyl]phenoxy]acetamide;hydrochloride | N-phenyl-2-[2-[[(phenylmethyl)amino]methyl]phenoxy]ethanamide;hydrochloride | SMR000144164 | cid_2962532
Type:
Small organic molecule
Emp. Form.:
C22H22N2O2
Mol. Mass.:
346.4223
SMILES:
O=C(COc1ccccc1CNCc1ccccc1)Nc1ccccc1
Structure:
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