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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48116
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
50000±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48116
Synonyms:
1,1-bis(oxidanylidene)-2-phenacyl-1,2-benzothiazol-3-one | 1,1-diketo-2-phenacyl-1,2-benzothiazol-3-one | 1,1-dioxo-2-phenacyl-1,2-benzothiazol-3-one | MLS000028285 | SMR000038129 | cid_658040
Type:
Small organic molecule
Emp. Form.:
C15H11NO4S
Mol. Mass.:
301.317
SMILES:
O=C(CN1C(=O)c2ccccc2S1(=O)=O)c1ccccc1
Structure:
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