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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM36894
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
24600±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM36894
Synonyms:
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide | MLS000038106 | SMR000040050 | cid_659101
Type:
Small organic molecule
Emp. Form.:
C15H10N2O2S
Mol. Mass.:
282.317
SMILES:
O=S1(=O)Nc2c(ccc3cccnc23)-c2ccccc12
Structure:
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