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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM34556
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
10000±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM34556
Synonyms:
2-(2-pyridinylmethylidene)-1-thiazolo[3,2-a]benzimidazolone | 2-(2-pyridylmethylene)thiazolo[3,2-a]benzimidazol-1-one | 2-(pyridin-2-ylmethylidene)-[1,3]thiazolo[3,2-a]benzimidazol-1-one | MLS000109246 | SMR000105191 | cid_722475
Type:
Small organic molecule
Emp. Form.:
C15H9N3OS
Mol. Mass.:
279.316
SMILES:
O=c1n2c(nc3ccccc23)sc1=Cc1ccccn1
Structure:
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