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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48242
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
310±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48242
Synonyms:
2-[4-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid methyl ester | 2-[4-[[(4-tert-butylphenyl)-oxomethyl]amino]phenyl]acetic acid methyl ester | MLS000535581 | SMR000143017 | cid_894181 | methyl 2-[4-[(4-tert-butylbenzoyl)amino]phenyl]acetate | methyl 2-[4-[(4-tert-butylphenyl)carbonylamino]phenyl]ethanoate | methyl {4-[(4-tert-butylbenzoyl)amino]phenyl}acetate
Type:
Small organic molecule
Emp. Form.:
C20H23NO3
Mol. Mass.:
325.4015
SMILES:
COC(=O)Cc1ccc(NC(=O)c2ccc(cc2)C(C)(C)C)cc1
Structure:
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