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Target
Zinc finger protein mex-5
Ligand
BDBM52776
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
66495±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52776
Synonyms:
MLS001029936 | N-[1-(3,4-Dimethoxy-phenyl)-eth-(E)-ylidene]-N'-(3-methyl-quinoxalin-2-yl)-hydrazine | N-[1-(3,4-dimethoxyphenyl)ethylideneamino]-3-methyl-2-quinoxalinamine | N-[1-(3,4-dimethoxyphenyl)ethylideneamino]-3-methyl-quinoxalin-2-amine | N-[1-(3,4-dimethoxyphenyl)ethylideneamino]-3-methylquinoxalin-2-amine | SMR000426953 | [1-(3,4-dimethoxyphenyl)ethylideneamino]-(3-methylquinoxalin-2-yl)amine | cid_2866692
Type:
Small organic molecule
Emp. Form.:
C19H20N4O2
Mol. Mass.:
336.3877
SMILES:
COc1ccc(cc1OC)C(C)N=Nc1nc2ccccc2nc1C |w:13.14|
Structure:
Search PDB for entries with ligand similarity: