Reaction Details Report a problem with these data
Target
POsterior Segregation
Ligand
BDBM53390
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
374±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM53390
Synonyms:
5-methyl-3-(phenyldiazenyl)pyrazolo[1,5-a]pyrimidine-2,7(1H,4H)-dione | 5-methyl-3-(phenylhydrazinylidene)-1H-pyrazolo[1,5-a]pyrimidine-2,7-dione | 5-methyl-3-(phenylhydrazono)-1H-pyrazolo[1,5-a]pyrimidine-2,7-quinone | MLS000325262 | SMR000161348 | cid_7309412
Type:
Small organic molecule
Emp. Form.:
C13H11N5O2
Mol. Mass.:
269.2587
SMILES:
Cc1cc(=O)n2[nH]c(=O)c(N=Nc3ccccc3)c2[nH]1 |w:10.9|
Structure:
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