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Target
Kallikrein-5
Ligand
BDBM32765
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
87.1±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM32765
Synonyms:
2-(benzotriazole-1-carbonyl)benzoic acid propargyl ester | 2-[1-benzotriazolyl(oxo)methyl]benzoic acid prop-2-ynyl ester | MLS000080837 | SMR000036164 | cid_658532 | prop-2-ynyl 2-(benzotriazol-1-ylcarbonyl)benzoate | prop-2-ynyl 2-(benzotriazole-1-carbonyl)benzoate
Type:
Small organic molecule
Emp. Form.:
C17H11N3O3
Mol. Mass.:
305.2875
SMILES:
O=C(OCC#C)c1ccccc1C(=O)n1nnc2ccccc12
Structure:
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