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Target
Delta-type opioid receptor
Ligand
BDBM62197
Substrate
n/a
Meas. Tech.
SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay
EC50
>32000±n/a nM
Citation
 PubChem, PC SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay PubChem Bioassay (2010)[AID] 
Target
Name:
Delta-type opioid receptor
Synonyms:
D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
40382.98
Organism:
Homo sapiens (Human)
Description:
Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor.
Residue:
372
Sequence:
MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM62197
Synonyms:
(phenylmethyl) N-[1-[(3-bromophenyl)carbamothioylamino]-2,2,2-tris(chloranyl)ethyl]carbamate | MLS-0425698.0001 | N-[1-[(3-bromophenyl)thiocarbamoylamino]-2,2,2-trichloro-ethyl]carbamic acid benzyl ester | N-[1-[[(3-bromoanilino)-sulfanylidenemethyl]amino]-2,2,2-trichloroethyl]carbamic acid (phenylmethyl) ester | benzyl N-[1-[(3-bromophenyl)carbamothioylamino]-2,2,2-trichloroethyl]carbamate | cid_3091269
Type:
Small organic molecule
Emp. Form.:
C17H15BrCl3N3O2S
Mol. Mass.:
511.648
SMILES:
ClC(Cl)(Cl)C(NC(=O)OCc1ccccc1)NC(=S)Nc1cccc(Br)c1
Structure:
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