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Target
Trans-activator protein BZLF1
Ligand
BDBM62431
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62431
Synonyms:
(5E)-3-benzyl-5-[(1,3-dimethyl-2-oxobenzimidazol-5-yl)methylidene]imidazolidine-2,4-dione | (5E)-3-benzyl-5-[(2-keto-1,3-dimethyl-benzimidazol-5-yl)methylene]hydantoin | (5E)-5-[(1,3-dimethyl-2-oxidanylidene-benzimidazol-5-yl)methylidene]-3-(phenylmethyl)imidazolidine-2,4-dione | (5E)-5-[(1,3-dimethyl-2-oxo-5-benzimidazolyl)methylidene]-3-(phenylmethyl)imidazolidine-2,4-dione | 3-benzyl-5-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)methylene]-2,4-imidazolidinedione | MLS000539109 | SMR000160447 | cid_1209501
Type:
Small organic molecule
Emp. Form.:
C20H18N4O3
Mol. Mass.:
362.3819
SMILES:
Cn1c2ccc(\C=C3\NC(=O)N(Cc4ccccc4)C3=O)cc2n(C)c1=O
Structure:
Search PDB for entries with ligand similarity: