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Target
Trans-activator protein BZLF1
Ligand
BDBM64844
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64844
Synonyms:
4-(3-chlorophenyl)sulfanyl-5-methoxy-2-pyridin-2-yl-pyrimidine | 4-(3-chlorophenyl)sulfanyl-5-methoxy-2-pyridin-2-ylpyrimidine | 4-[(3-chlorophenyl)sulfanyl]-2-(2-pyridinyl)-5-pyrimidinyl methyl ether | 4-[(3-chlorophenyl)thio]-5-methoxy-2-(2-pyridinyl)pyrimidine | 4-[(3-chlorophenyl)thio]-5-methoxy-2-(2-pyridyl)pyrimidine | MLS000325791 | SMR000169707 | cid_3740241
Type:
Small organic molecule
Emp. Form.:
C16H12ClN3OS
Mol. Mass.:
329.804
SMILES:
COc1cnc(nc1Sc1cccc(Cl)c1)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: