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Target
Trans-activator protein BZLF1
Ligand
BDBM45140
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM45140
Synonyms:
2-(3,5-dimethyl-1-pyrazolyl)-N-[(4-methoxyphenyl)methylideneamino]-6-methyl-4-pyrimidinamine | 2-(3,5-dimethylpyrazol-1-yl)-N-[(4-methoxyphenyl)methylideneamino]-6-methyl-pyrimidin-4-amine | 2-(3,5-dimethylpyrazol-1-yl)-N-[(4-methoxyphenyl)methylideneamino]-6-methylpyrimidin-4-amine | MLS000589393 | N-[2-(3,5-Dimethyl-pyrazol-1-yl)-6-methyl-pyrimidin-4-yl]-N'-[1-(4-methoxy-phenyl)-meth-(E)-ylidene]-hydrazine | SMR000212741 | [2-(3,5-dimethylpyrazol-1-yl)-6-methyl-pyrimidin-4-yl]-(p-anisylideneamino)amine | cid_5093634
Type:
Small organic molecule
Emp. Form.:
C18H20N6O
Mol. Mass.:
336.391
SMILES:
COc1ccc(CN=Nc2cc(C)nc(n2)-n2nc(C)cc2C)cc1 |w:8.8|
Structure:
Search PDB for entries with ligand similarity: