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Target
Trans-activator protein BZLF1
Ligand
BDBM64849
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64849
Synonyms:
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-keto-N-[4-(2-pyridyl)thiazol-2-yl]pyrrolidine-3-carboxamide | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxidanylidene-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)pyrrolidine-3-carboxamide | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)pyrrolidine-3-carboxamide | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxo-N-[4-(2-pyridinyl)-2-thiazolyl]-3-pyrrolidinecarboxamide | MLS000394395 | SMR000261836 | cid_5033819
Type:
Small organic molecule
Emp. Form.:
C21H18N4O4S
Mol. Mass.:
422.457
SMILES:
O=C(Nc1nc(cs1)-c1ccccn1)C1CN(C(=O)C1)c1ccc2OCCOc2c1
Structure:
Search PDB for entries with ligand similarity: