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Target
Bcl-2-like protein 11
Ligand
BDBM67047
Substrate
n/a
Meas. Tech.
Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis
EC50
>350000±n/a nM
Citation
 PubChem, PC Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis PubChem Bioassay (2010)[AID] 
Target
Name:
Bcl-2-like protein 11
Synonyms:
B2L11_HUMAN | BCL2-like 11 isoform 1 | BCL2L11 | BIM
Type:
PROTEIN
Mol. Mass.:
22175.26
Organism:
Homo sapiens (Human)
Description:
EBI_101325
Residue:
198
Sequence:
MAKQPSDVSSECDREGRQLQPAERPPQLRPGAPTSLQTEPQGNPEGNHGGEGDSCPHGSPQGPLAPPASPGPFATRSPLFIFMRRSSLLSRSSSGYFSFDTDRSPAPMSCDKSTQTPSPPCQAFNHYLSAMASMRQAEPADMRPEIWIAQELRRIGDEFNAYYARRVFLNNYQAAEDHPRMVILRLLRYIVRLVWRMH
  
Inhibitor
Name:
BDBM67047
Synonyms:
6-keto-1-phenyl-4,5-dihydropyridazine-3-carboxylic acid [2-(4,5-dimethyl-2-nitro-anilino)-2-keto-ethyl] ester | 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylic acid [2-(4,5-dimethyl-2-nitroanilino)-2-oxoethyl] ester | MLS002248940 | SMR001316395 | [2-(4,5-dimethyl-2-nitroanilino)-2-oxoethyl] 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylate | [2-[(4,5-dimethyl-2-nitro-phenyl)amino]-2-oxidanylidene-ethyl] 6-oxidanylidene-1-phenyl-4,5-dihydropyridazine-3-carboxylate | cid_4290049
Type:
Small organic molecule
Emp. Form.:
C21H20N4O6
Mol. Mass.:
424.4067
SMILES:
Cc1cc(NC(=O)COC(=O)[C+]2CCC(=O)N([N-]2)c2ccccc2)c(cc1C)[N+]([O-])=O
Structure:
Search PDB for entries with ligand similarity: