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Target
Bcl-2-like protein 11
Ligand
BDBM67058
Substrate
n/a
Meas. Tech.
Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis
EC50
>350000±n/a nM
Citation
 PubChem, PC Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis PubChem Bioassay (2010)[AID] 
Target
Name:
Bcl-2-like protein 11
Synonyms:
B2L11_HUMAN | BCL2-like 11 isoform 1 | BCL2L11 | BIM
Type:
PROTEIN
Mol. Mass.:
22175.26
Organism:
Homo sapiens (Human)
Description:
EBI_101325
Residue:
198
Sequence:
MAKQPSDVSSECDREGRQLQPAERPPQLRPGAPTSLQTEPQGNPEGNHGGEGDSCPHGSPQGPLAPPASPGPFATRSPLFIFMRRSSLLSRSSSGYFSFDTDRSPAPMSCDKSTQTPSPPCQAFNHYLSAMASMRQAEPADMRPEIWIAQELRRIGDEFNAYYARRVFLNNYQAAEDHPRMVILRLLRYIVRLVWRMH
  
Inhibitor
Name:
BDBM67058
Synonyms:
5,6-dimethoxy-2-(4-methylsulfonylphenyl)-N-(4-oxidanylbutyl)-1-benzothiophene-3-carboxamide | MLS002473592 | N-(4-hydroxybutyl)-2-(4-mesylphenyl)-5,6-dimethoxy-benzothiophene-3-carboxamide | N-(4-hydroxybutyl)-5,6-dimethoxy-2-(4-methylsulfonylphenyl)-1-benzothiophene-3-carboxamide | SMR001397759 | cid_44202239
Type:
Small organic molecule
Emp. Form.:
C22H25NO6S2
Mol. Mass.:
463.567
SMILES:
COc1cc2sc(c(C(=O)NCCCCO)c2cc1OC)-c1ccc(cc1)S(C)(=O)=O
Structure:
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