Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM51208
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
690.35±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM51208
Synonyms:
(4-nitrobenzofurazan-5-yl)amine | 4-nitro-2,1,3-benzoxadiazol-5-amine | MLS000728227 | SMR000306920 | cid_555700
Type:
Small organic molecule
Emp. Form.:
C6H4N4O3
Mol. Mass.:
180.121
SMILES:
Nc1ccc2nonc2c1[N+]([O-])=O
Structure:
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