Reaction Details Report a problem with these data
Target
Hyaluronidase-1
Ligand
BDBM81861
Substrate
n/a
Meas. Tech.
Stains-all Assay
pH
7±0
Temperature
310.15±0 K
IC50
3.321e+4±n/a nM
Citation
Olgen, S; Kaessler, A; Nebioglu, D; Jose, J New potent indole derivatives as hyaluronidase inhibitors. Chem Biol Drug Des 70:547-51 (2007) [PubMed] Article
More Info.:
Target
Name:
Hyaluronidase-1
Synonyms:
HYAL1 | HYAL1_HUMAN | Hyaluronidase | Hyaluronidase-1 | Hyaluronoglucosaminidase-1 | LUCA1
Type:
Protein
Mol. Mass.:
48369.09
Organism:
Homo sapiens (Human)
Description:
Q1279
Residue:
435
Sequence:
MAAHLLPICALFLTLLDMAQGFRGPLLPNRPFTTVWNANTQWCLERHGVDVDVSVFDVVANPGQTFRGPDMTIFYSSQLGTYPYYTPTGEPVFGGLPQNASLIAHLARTFQDILAAIPAPDFSGLAVIDWEAWRPRWAFNWDTKDIYRQRSRALVQAQHPDWPAPQVEAVAQDQFQGAARAWMAGTLQLGRALRPRGLWGFYGFPDCYNYDFLSPNYTGQCPSGIRAQNDQLGWLWGQSRALYPSIYMPAVLEGTGKSQMYVQHRVAEAFRVAVAAGDPNLPVLPYVQIFYDTTNHFLPLDELEHSLGESAAQGAAGVVLWVSWENTRTKESCQAIKEYMDTTLGPFILNVTSGALLCSQALCSGHGRCVRRTSHPKALLLLNPASFSIQLTPGGGPLSLRGALSLEDQAQMAVEFKCRCYPGWQAPWCERKSMW