Reaction Details Report a problem with these data
Target
Beta-arrestin-2
Ligand
BDBM81875
Substrate
n/a
Ki
154.88±n/a nM
Comments
PDSP_831
Citation
Wong, DT; Threlkeld, PG; Robertson, DW Affinities of fluoxetine, its enantiomers, and other inhibitors of serotonin uptake for subtypes of serotonin receptors. Neuropsychopharmacology 5:43-7 (1991) [PubMed]
More Info.:
Target
Name:
Beta-arrestin-2
Synonyms:
5-HT2C | ARRB2 | ARRB2_BOVIN | Beta-arrestin-2 | HTR2C
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47232.00
Organism:
Beef
Description:
5-HT2C HTR2C Beef::P32120
Residue:
420
Sequence:
MGEKPGTRVFKKSSPNCKLTVYLGKRDFVDHLDKVDPVDGVVLVDPDYLKDRKVFVTLTCAFRYGREDLDVLGLSFRKDLFIANYQAFPPTPNPPRPPTRLQERLLRKLGQHAHPFFFTIPQNLPCSVTLQPGPEDTGKACGVDFEIRAFCAKSLEEKSHKRNSVRLVIRKVQFAPEKPGPQPSAETTRHFLMSDRSLHLEASLDKELYYHGEPLNVNVHVTNNSTKTVKKIKVSVRQYADICLFSTAQYKCPVAQVEQDDQVSPSSTFCKVYTITPLLSNNREKRGLALDGKLKHEDTNLASSTIVKEGANKEVLGILVSYRVKVKLVVSRGGDVSVELPFVLMHPKPHDHIALPRPQSAATHPPTLLPSAVPETDAPVDTNLIEFETNYATDDDIVFEDFARLRLKGLKDEDYDDQFC