Reaction Details
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5-hydroxytryptamine receptor 2B
Ligand
BDBM81966
Substrate
n/a
Ki
125±n/a nM
Comments
PDSP_710
Citation
McKenna, DJ; Peroutka, SJ Differentiation of 5-hydroxytryptamine2 receptor subtypes using 125I-R-(-)2,5-dimethoxy-4-iodo-phenylisopropylamine and 3H-ketanserin. J Neurosci 9:3482-90 (1989) [PubMed] More Info.:
Target
Name:
5-hydroxytryptamine receptor 2B
Synonyms:
5-HT2B | 5-hydroxytryptamine 2B receptor | HTR2B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
15564.62
Organism:
BOVINE
Description:
Q8MI09
Residue:
137
Sequence:
KPPQRLTWLTVSTVFQRDETPCSSPEKVAMLDGFHKDKTLPNASADILMRRMSTVGKKSVQTISNEQRASKVLGIVFFLFLLMWCPFFITNVTLVLCDSCNQTTLNMLLEIFVWIGYVSSGVNPLVYTLFNKTFRDA
Inhibitor
Name:
BDBM81966
Synonyms:
DOB,S(+)
Type:
n/a
Emp. Form.:
C19H18N2O6
Mol. Mass.:
370.356
SMILES:
COC(CO)C(=O)O[C@@H](C)c1cccc2nc3c(cccc3nc12)C(O)=O |r|
Structure:
