Reaction Details Report a problem with these data
Target
Inner capsid protein sigma-2
Ligand
BDBM82273
Substrate
n/a
Ki
15.84±n/a nM
Comments
PDSP_1621
Citation
Hegde, SS; Bonhaus, DW; Johnson, LG; Leung, E; Clark, RD; Eglen, RM RS 39604: a potent, selective and orally active 5-HT4 receptor antagonist. Br J Pharmacol 115:1087-95 (1995) [PubMed] Article
More Info.:
Target
Name:
Inner capsid protein sigma-2
Synonyms:
S2 | SIGM2_REOVL | Sigma-2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47118.43
Organism:
Reovirus type 1 (strain Lang) (T1L) (Mammalian orthoreovirus 1)
Description:
P11314
Residue:
418
Sequence:
MARAAFLFKTVGFGGLQNVPINDELSSHLLRAGNSPWQLTQFLDWISLGRGLATSALVPTAGSRYYQMSCLLSGTLQIPFRPNHRWGDIRFLRLVWSAPTLDGLVVAPPQVLAQPALQAQADRVYDCDDYPFLARDPRFKHRVYQQLSAVTLLNLTGFGPISYVRVDEDMWSGDVNQLLMNYFGHTFAEIAYTLCQASANRPWEHDGTYARMTQIILSLFWLSYVGVIHQQNTYRTFYFQCNRRGDAAEVWILSCSLNHSAQIRPGNRSLFVMPTSPDWNMDVNLILSSTLTGCLCSGSQLPLIDNNSVPAVSRNIHGWTGRAGNQLHGFQVRRMVTEFCDRLRRDGVMTQAQQNQIEALADQTQQFKRDKLEAWAREDDQYNQANPNSTMFRTKPFTNAQWGRGNTGATSAAIAALI