Reaction Details Report a problem with these data
Target
Beta-arrestin-1
Ligand
BDBM82381
Substrate
n/a
Ki
0.51±n/a nM
Comments
PDSP_1054
Citation
Hwang, SB; Lam, MH; Alberts, AW; Bugianesi, RL; Chabala, JC; Ponpipom, MM Biochemical and pharmacological characterization of L-659,989: an extremely potent, selective and competitive receptor antagonist of platelet-activating factor. J Pharmacol Exp Ther 246:534-41 (1988) [PubMed]
More Info.:
Target
Name:
Beta-arrestin-1
Synonyms:
ARRB1 | ARRB1_RABIT | Beta-arrestin-1 | Cholinergic, muscarinic | OPIATE Delta | PAF Platelet activating factor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
46360.54
Organism:
RABBIT
Description:
Cholinergic, muscarinic 0 RABBIT::Q95223
Residue:
410
Sequence:
MGDKGTRVFKKASPNGKLTVYLGKRGFVDHIDLVDPVDGVVLVDPEYLKERRVYVTLTCAFRYGREDLDVLGLTFRKDLFVANVQSFPPAPEDKKPLTRLQERLIKKLGEHAYPFTFEIPPKLPCSVTLQPGPEDTGKACGVDYEVKAFCAENLEEKIHKRNSVRLVIRKVQYAPERPGPHPTAETTRLFLMSDKPLHLEASLDKEIYYHGEPIIVNVHVTNNTNKTVKKIKISVRQYADICLFNTAQYKCPVAMEEADDTVAPSSTFCKVYTLTPFLANNREKRGLALDGKLKHEDTNLASSTLMREGANREILGIIVSYKVKVKLVVSRGGDVAVELPFTLMHPKPKEEPPHREVPENETPVDTNLIELDTNDDDIVFEDFARQRLKGMKDDKEEEDDVTGSPRLNDR