Target
Neuropeptide Y receptor type 2
Ligand
BDBM82287
Substrate
n/a
Ki
2.34±n/a nM
Comments
PDSP_1389
Citation
 Gerald, CAdham, NKao, HTOlsen, MALaz, TMSchechter, LEBard, JAVaysse, PJHartig, PRBranchek, TA The 5-HT4 receptor: molecular cloning and pharmacological characterization of two splice variants. EMBO J 14:2806-15 (1995) [PubMed] 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM82287
Synonyms:
NPY2-36 | NPY2-36, human | NPY2-36, porcine
Type:
Small organic molecule
Emp. Form.:
C181H278N54O55
Mol. Mass.:
4090.4728
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: