Reaction Details Report a problem with these data
Target
Pituitary adenylate cyclase-activating polypeptide
Ligand
BDBM82446
Substrate
n/a
Ki
10±n/a nM
Comments
PDSP_2420
Citation
 Hou, X; Vandermeers, A; Gourlet, P; Vandermeers-Piret, MC; Robberecht, P Structural requirements for the occupancy of rat brain PACAP receptors and adenylate cyclase activation. Neuropharmacology 33:1189-95 (1994) [PubMed]  Article 
Target
Name:
Pituitary adenylate cyclase-activating polypeptide
Synonyms:
Adcyap1 | PACAP | PACAP-27 | PACAP-38 | PACA_RAT | Pituitary adenylate cyclase-activating polypeptide
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19565.66
Organism:
RAT
Description:
PACAP 0 RAT::P13589
Residue:
175
Sequence:
MTMCSGARLALLVYGIIMHNSVSCSPAAGLSFPGIRPEEEAYDQDGNPLQDFYDWDPPGAGSPASALRDAYALYYPADRRDVAHEILNEAYRKVLDQLSARKYLQSMVARGMGENLAAAAVDDRAPLTKRHSDGIFTDSYSRYRKQMAVKKYLAAVLGKRYKQRVKNKGRRIAYL
  
Inhibitor
Name:
BDBM82446
Synonyms:
[DArg2]PACAP(1-38)
Type:
Small organic molecule
Emp. Form.:
C205H345N69O52S
Mol. Mass.:
4640.429
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: