Reaction Details Report a problem with these data
Target
Melatonin receptor
Ligand
BDBM50043289
Substrate
n/a
Ki
4±n/a nM
Comments
PDSP_7419
Citation
 Morgan, PJ; Barrett, P; Howell, HE; Helliwell, R Melatonin receptors: localization, molecular pharmacology and physiological significance. Neurochem Int 24:101-46 (1994) [PubMed]  Article 
Target
Name:
Melatonin receptor
Synonyms:
Melatonin | Melatonin receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13287.02
Organism:
RABBIT
Description:
Q9BE38
Residue:
114
Sequence:
MIWMLTLVAVMPNLHTGTLQYDPRVYSCTFSQSVSSAYTIAVVVFHFIIPMLMSSCCYLRIWILVLQVRRRVKPDNKPKLKPQDFRNFITMFVVFVLFAICWAPLNFIVLLGRS
  
Inhibitor
Name:
BDBM50043289
Synonyms:
CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-yl)-ethyl]-acetamide | N-[2-(6-Chloro-5-methoxy-1H-indol-3-yl)-ethyl]-acetamide(6-Chloromelatonin) | melatonin, 6-Chloro
Type:
Small organic molecule
Emp. Form.:
C13H15ClN2O2
Mol. Mass.:
266.723
SMILES:
COc1cc2c(CCNC(C)=O)c[nH]c2cc1Cl
Structure:
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