Reaction Details Report a problem with these data
Target
Somatostatin receptor type 2
Ligand
BDBM84641
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_1946
Citation
 Raynor, K; Murphy, WA; Coy, DH; Taylor, JE; Moreau, JP; Yasuda, K; Bell, GI; Reisine, T Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides. Mol Pharmacol 43:838-44 (1993) [PubMed] 
Target
Name:
Somatostatin receptor type 2
Synonyms:
SOMATOSTATIN SST2 | SSR2_MOUSE | Smstr2 | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sst2 | Sstr2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41234.26
Organism:
MOUSE
Description:
SOMATOSTATIN SST2 SSTR2 MOUSE::P30875
Residue:
369
Sequence:
MEMSSEQLNGSQVWVSSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCGNTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMTVDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWCVSLLVILPIMIYAGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGIRVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVILTYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTEDGERSDSKQDKSRLNETTETQRTLLNGDLQTSI
  
Inhibitor
Name:
BDBM84641
Synonyms:
SA V | c[Aoc-Phe-D-Trp-Lys-Thr(Bzl)]
Type:
Small organic molecule
Emp. Form.:
C46H62N8O6
Mol. Mass.:
823.0345
SMILES:
CC(OCc1ccccc1)C1NC(=O)C(CCCCCCCCN)NC(=O)C(Cc2ccccc2)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(CCCN)NC1=O
Structure:
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