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Target
G-protein coupled receptor 52
Ligand
BDBM50252187
Substrate
n/a
Meas. Tech.
ChEBML_1684383
EC50
83±n/a nM
Citation
 Tokumaru, K; Ito, Y; Nomura, I; Nakahata, T; Shimizu, Y; Kurimoto, E; Aoyama, K; Aso, K Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists. Bioorg Med Chem 25:3098-3115 (2017) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 52
Synonyms:
GPR52 | GPR52_HUMAN | Probable G-protein coupled receptor 52
Type:
PROTEIN
Mol. Mass.:
41366.15
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108391
Residue:
361
Sequence:
MNESRWTEWRILNMSSGIVNVSERHSCPLGFGHYSVVDVCIFETVVIVLLTFLIIAGNLTVIFVFHCAPLLHHYTTSYFIQTMAYADLFVGVSCLVPTLSLLHYSTGVHESLTCQVFGYIISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIILIWIYSCLIFLPSFFGWGKPGYHGDIFEWCATSWLTSAYFTGFIVCLLYAPAAFVVCFTYFHIFKICRQHTKEINDRRARFPSHEVDSSRETGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSFLTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCMCVKDQEAQEPKPRKRANSCSI
  
Inhibitor
Name:
BDBM50252187
Synonyms:
CHEMBL4099668
Type:
Small organic molecule
Emp. Form.:
C21H19F3N2OS
Mol. Mass.:
404.449
SMILES:
CCc1cc(ccc1C(N)=O)-c1sc(Cc2cccc(c2)C(F)(F)F)nc1C
Structure:
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