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TargetAdenosine A2b receptor
LigandBDBM50455533
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1754702
Ki 1.3±n/a nM
Citation Köse, MGollos, SKarcz, TFiene, AHeisig, FBehrenswerth, AKie?-Kononowicz, KNamasivayam, VMüller, CE Fluorescent-Labeled Selective Adenosine A J Med Chem61:4301-4316 (2018) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Adenosine A2b receptor
Name:Adenosine A2b receptor
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:36130.09
Organism:Mus musculus
Description:ChEMBL_11831
Residue:332
Sequence:
MQLETQDALYVALELVIAALAVAGNVLVCAAVGASSALQTPTNYFLVSLATADVAVGLFA
IPFAITISLGFCTDFHGCLFLACFVLVLTQSSIFSLLAVAVDRYLAIRVPLRYKGLVTGT
RARGIIAVLWVLAFGIGLTPFLGWNSKDSATSNCTELGDGIANKSCCPVTCLFENVVPMS
YMVYFNFFGCVLPPLLIMLVIYIKIFMVACKQLQRMELMDHSRTTLQREIHAAKSLAMIV
GIFALCWLPVHAINCITLFHPALAKDKPKWVMNVAILLSHANSVVNPIVYAYRNRDFRYS
FHKIISRYVLCQAETKGGSGQAGAQSTLSLGL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50455533
NameBDBM50455533
Synonyms:CHEMBL4205635
TypeSmall organic molecule
Emp. Form.C31H34BF2N7O4
Mol. Mass.617.454
SMILESCCCn1c(=O)[nH]c2nc([nH]c2c1=O)-c1ccc(OCC(=O)NCCC2=C3C(C)=CC(C)=[N+]3[B-](F)(F)n3c(C)cc(C)c23)cc1 |c:27,30,33|
Structure
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n/a