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Target
Glucose-dependent insulinotropic receptor
Ligand
BDBM29080
Substrate
n/a
Meas. Tech.
ChEMBL_1778942 (CHEMBL4235934)
EC50
3200±n/a nM
Citation
 Fang, Y; Xu, J; Li, Z; Yang, Z; Xiong, L; Jin, Y; Wang, Q; Xie, S; Zhu, W; Chang, S Design and synthesis of novel pyrimido[5,4-d]pyrimidine derivatives as GPR119 agonist for treatment of type 2 diabetes. Bioorg Med Chem 26:4080-4087 (2018) [PubMed]  Article 
Target
Name:
Glucose-dependent insulinotropic receptor
Synonyms:
G-protein coupled receptor 119 (GPR119) | GP119_HUMAN | GPR119 | Glucose-dependent insulinotropic receptor
Type:
Protein
Mol. Mass.:
36901.49
Organism:
Homo sapiens (Human)
Description:
Q8TDV5
Residue:
335
Sequence:
MESSFSFGVILAVLASLIIATNTLVAVAVLLLIHKNDGVSLCFTLNLAVADTLIGVAISGLLTDQLSSPSRPTQKTLCSLRMAFVTSSAAASVLTVMLITFDRYLAIKQPFRYLKIMSGFVAGACIAGLWLVSYLIGFLPLGIPMFQQTAYKGQCSFFAVFHPHFVLTLSCVGFFPAMLLFVFFYCDMLKIASMHSQQIRKMEHAGAMAGGYRSPRTPSDFKALRTVSVLIGSFALSWTPFLITGIVQVACQECHLYLVLERYLWLLGVGNSLLNPLIYAYWQKEVRLQLYHMALGVKKVLTSFLLFLSARNCGPERPRESSCHIVTISSSEFDG
  
Inhibitor
Name:
BDBM29080
Synonyms:
CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA | Oleoyl monoethanolamide | Oleoylethanolamide (OEA)
Type:
n/a
Emp. Form.:
C20H39NO2
Mol. Mass.:
325.5292
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)NCCO
Structure:
Search PDB for entries with ligand similarity: