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Target
Proteasome subunit beta type-9
Ligand
BDBM50464981
Substrate
n/a
Meas. Tech.
ChEMBL_1783551 (CHEMBL4255068)
IC50
10600±n/a nM
Citation
Richy, N; Sarraf, D; Maréchal, X; Janmamode, N; Le Guével, R; Genin, E; Reboud-Ravaux, M; Vidal, J Structure-based design of human immuno- and constitutive proteasomes inhibitors. Eur J Med Chem 145:570-587 (2018) [PubMed] Article
More Info.:
Target
Name:
Proteasome subunit beta type-9
Synonyms:
LMP2 | Low molecular mass protein 2 | Macropain chain 7 | Multicatalytic endopeptidase complex chain 7 | PSB9_HUMAN | PSMB6i | PSMB9 | Proteasome chain 7 | Proteasome subunit beta-1i | RING12 | Really interesting new gene 12 protein
Type:
PROTEIN
Mol. Mass.:
23256.49
Organism:
Human
Description:
ChEMBL_106197
Residue:
219
Sequence:
MLRAGAPTGDLPRAGEVHTGTTIMAVEFDGGVVMGSDSRVSAGEAVVNRVFDKLSPLHERIYCALSGSAADAQAVADMAAYQLELHGIELEEPPLVLAAANVVRNISYKYREDLSAHLMVAGWDQREGGQVYGTLGGMLTRQPFAIGGSGSTFIYGYVDAAYKPGMSPEECRRFTTDAIALAMSRDGSSGGVIYLVTITAAGVDHRVILGNELPKFYDE