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Target
Muscarinic receptor M1
Ligand
BDBM50035991
Substrate
n/a
Meas. Tech.
ChEMBL_140162 (CHEMBL745467)
Ki
36±n/a nM
Citation
 Kiesewetter, DO; Lee, J; Lang, L; Park, SG; Paik, CH; Eckelman, WC Preparation of 18F-labeled muscarinic agonist with M2 selectivity. J Med Chem 38:5-8 (1995) [PubMed]  Article 
Target
Name:
Muscarinic receptor M1
Synonyms:
Muscarinic acetylcholine receptor M1
Type:
PROTEIN
Mol. Mass.:
15022.43
Organism:
Bos taurus
Description:
ChEMBL_140161
Residue:
139
Sequence:
ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYSWKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKGRERAGKGQKPRGKEQLAKR
  
Inhibitor
Name:
BDBM50035991
Synonyms:
1-Methyl-4-(4-pentylsulfanyl-[1,2,5]thiadiazol-3-yl)-1,2,3,6-tetrahydro-pyridine | CHEMBL350332
Type:
Small organic molecule
Emp. Form.:
C13H21N3S2
Mol. Mass.:
283.456
SMILES:
CCCCCSc1nsnc1C1=CCN(C)CC1 |t:12|
Structure:
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