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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50006975
Substrate/Competitorn/a
Meas. Tech.ChEMBL_200976
Ki 12±n/a nM
Citation Glennon, RAAblordeppey, SYIsmaiel, AMel-Ashmawy, MBFischer, JBHowie, KB Structural features important for sigma 1 receptor binding. J Med Chem37:1214-9 (1994) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma opioid receptor
Synonyms:Aging-associated gene 8 protein | SIG-1R | SR-BP | SR31747-binding protein | Sigma 1-type opioid receptor | Sigma opioid receptor | Sigma1R | hSigmaR1
Type:Enzyme Catalytic Domain
Mol. Mass.:25124.85
Organism:Homo sapiens (Human)
Description:Sigma 0 HUMAN::Q99720
Residue:223
Sequence:
MQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQDP
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BDBM50006975
NameBDBM50006975
Synonyms:CHEMBL19802 | [2-(4-Bromo-phenyl)-1-methyl-ethyl]-(3-phenyl-propyl)-amine
TypeSmall organic molecule
Emp. Form.C18H22BrN
Mol. Mass.332.278
SMILESCC(Cc1ccc(Br)cc1)NCCCc1ccccc1
Structure
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