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Target
D(3) dopamine receptor
Ligand
BDBM50496575
Substrate
n/a
Meas. Tech.
ChEMBL_1299394 (CHEMBL3136929)
Ki
0.900000±n/a nM
Citation
 Tu, Z; Li, S; Li, A; Taylor, M; Ho, D; Malik, M; Luedtke, RR; Mach, RH Synthesis and  Medchemcomm 4:1283-1289 (2013) [PubMed]  Article 
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3
Type:
n/a
Mol. Mass.:
44243.43
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
400
Sequence:
MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTVCSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQQTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRKLSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHVSPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
  
Inhibitor
Name:
BDBM50496575
Synonyms:
CHEMBL3133870
Type:
Small organic molecule
Emp. Form.:
C27H33FN4O6
Mol. Mass.:
528.5725
SMILES:
OC(=O)C(O)=O.FCCOc1ccccc1N1CCN(CCCCNC(=O)c2c[nH]c3ccccc23)CC1
Structure:
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